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科研机构
上海药物研究所 [23]
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期刊论文 [23]
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2021 [2]
2019 [1]
2018 [4]
2016 [2]
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Rosmarinic Acid Suppresses Abdominal Aortic Aneurysm Progression in Apolipoprotein E-deficient Mice
期刊论文
PLANTA MEDICA, 2021, 页码: 14
作者:
Bian, Huimiao
;
Wang, Yang
;
Wu, Peng
;
Han, Na
;
Wang, Linlin
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2021/12/16
abdominal aortic aneurysm
rosmarinic acid
salvianolic acid C
salvianolic acid B
Salvia miltiorrhiza Bunge
Labiatae
PRMT1 is a novel molecular therapeutic target for clear cell renal cell carcinoma
期刊论文
THERANOSTICS, 2021, 卷号: 11, 期号: 11, 页码: 5387-5403
作者:
Wang, Jianfeng
;
Wang, Chen
;
Xu, Pan
;
Li, Xiao
;
Lu, Yongning
收藏
  |  
浏览/下载:130/0
  |  
提交时间:2021/05/24
clear cell renal cell carcinoma
protein arginine methyltransferase 1
therapeutic
lipocalin2 (LCN2)
sunitinib
Discovery of trisubstituted nicotinonitrile derivatives as novel human GCN5 inhibitors through AlphaScreen-based high throughput screening
期刊论文
RSC ADVANCES, 2019, 卷号: 9, 期号: 9, 页码: 4917-4924
作者:
Tao, Hongru
;
Wang, Jun
;
Lu, Wenchao
;
Zhang, Rukang
;
Xie, Yiqian
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/07/01
Targeting AKT with Oridonin Inhibits Growth of Esophageal Squamous Cell Carcinoma In Vitro and Patient-Derived Xenografts In Vivo
期刊论文
MOLECULAR CANCER THERAPEUTICS, 2018, 卷号: 17, 期号: 7, 页码: 1540-1553
作者:
Song, Mengqiu
;
Liu, Xuejiao
;
Liu, Kangdong
;
Zhao, Ran
;
Huang, Hai
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2019/01/08
Discovery of 1,8-acridinedione derivatives as novel GCN5 inhibitors via high throughput screening
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 151, 页码: 740-751
作者:
Xiong, Huan
;
Han, Jie
;
Wang, Jun
;
Lu, Wenchao
;
Wang, Chen
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
Epigenetics
Histone acetyltransferase
GCN5
High throughput screening
1,8-Acridinedione derivative
Identification and Characterizations of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Scaffold Hopping- and 2D-Molecular Fingerprint-Based Similarity Search
期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 3
作者:
Ding, Hong
;
Lu, Wen Chao
;
Hu, Jun Chi
;
Liu, Yu-Chih
;
Zhang, Chen Hua
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2019/01/08
SET7
inhibitor
similarity search
ligand-based drug design
chemical biology probe
7 alpha,8 alpha-Epoxynagilactones and their glucosides from the twigs of Podocarpus nagi: Isolation, structures, and cytotoxic activities
期刊论文
FITOTERAPIA, 2018, 卷号: 125, 页码: 174-183
作者:
Zheng, Yuan-Dong
;
Bai, Gang
;
Tang, Chunping
;
Ke, Chang-Qiang
;
Yao, Sheng
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
Podocarpus nagi
Type B nagilactone
Cytotoxic activity
Apoptosis
Proteasome Inhibition Contributed to the Cytotoxicity of Arenobufagin after Its Binding with Na, K-ATPase in Human Cervical Carcinoma HeLa Cells
期刊论文
PLOS ONE, 2016, 卷号: 11, 期号: 7
作者:
Yue, Qingxi
;
Zhen, Hong
;
Huang, Ming
;
Zheng, Xi
;
Feng, Lixing
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
Metabolomics study on the antitumor effect of marine natural compound flexibilide in HCT-116 colon cancer cell line
期刊论文
JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 2016, 卷号: 1014, 页码: 17-23
作者:
Gao, Dan
;
Wang, Yini
;
Xie, Weiyi
;
Yang, Ti
;
Jiang, Yuyang
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
Metabolomics
UPLC/Q-TOF MS
Flexibilide
HCT-116 cells
Action mechanism
Synthesis and Biological Activities of Novel 2,5-Disubstituted-1,3,4-thiadiazole Derivatives
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2015, 卷号: 35, 期号: 1, 页码: 129-136
作者:
Li Yingjun
;
Yu Yang
;
Jin Kun
;
Gao Lixin
;
Luo Tongchuan
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
2,5-disubstituted-1,3,4-thiadiazole
benzisoselenazolone
synthesis
bioactivity
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