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科研机构
上海药物研究所 [25]
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期刊论文 [25]
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2020 [3]
2018 [2]
2017 [1]
2012 [1]
2011 [2]
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Molecular insights into the human CLC-7/Ostm1 transporter
期刊论文
SCIENCE ADVANCES, 2020, 卷号: 6, 期号: 33, 页码: 10
作者:
Zhang, Sensen
;
Liu, Yang
;
Zhang, Bing
;
Zhou, Jun
;
Li, Tianyu
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/12/24
Discovery of aryl sulfonamide-selective Nav1.7 inhibitors with a highly hydrophobic ethanoanthracene core
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 293-302
作者:
Wang, Jin-tao
;
Zheng, Yue-ming
;
Chen, Yue-ting
;
Gu, Min
;
Gao, Zhao-bing
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2020/07/01
Nav1
7 sodium channel
aryl sulfonamide
maprotiline
compound 10o
electrophysiology
acetic acid-induced visceral pain
analgesic activity
discoveryofarylsulfonamideselectivenav17inhibitorswithahighlyhydrophobicethanoanthracenecore
期刊论文
actapharmacologicasinica, 2020, 卷号: 41, 期号: 3, 页码: 293
作者:
Wang Jintao
;
Zheng Yueming
;
Chen Yueting
;
Gu Min
;
Gao Zhaobing
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/07/01
Nav1.7 sodium channel
aryl sulfonamide
maprotiline
compound 10o
electrophysiology
acetic acid-induced visceral pain
analgesic activity
Enhancing inactivation rather than reducing activation of Nav1.7 channels by a clinically effective analgesic CNV1014802
期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 4, 页码: 587-596
作者:
Zheng, Yue-ming
;
Wang, Wan-fu
;
Li, Yan-fen
;
Yu, Yong
;
Gao, Zhao-bing
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2019/01/08
Nav1.7 channels
analgesics
CNV1014802
inactivated state
paroxysmal extreme pain disorder
A Statistical Thermodynamic Model for Ligands Interacting With Ion Channels: Theoretical Model and Experimental Validation of the KCNQ2 Channel
期刊论文
FRONTIERS IN PHARMACOLOGY, 2018, 卷号: 9
作者:
Bai, Fang
;
Pi, Xiaoping
;
Li, Ping
;
Zhou, Pingzheng
;
Yang, Huaiyu
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
KCNQ2 potassium channel
hill equation
thermodynamic model
patch clamp electrophysiology
activators
An allosteric ligand-binding site in the extracellular cap of K2P channels
期刊论文
NATURE COMMUNICATIONS, 2017, 卷号: 8
作者:
Luo, Qichao
;
Chen, Liping
;
Cheng, Xi
;
Ma, Yuqin
;
Li, Xiaona
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
Structure and molecular mechanism of an anion-selective mechanosensitive channel of small conductance
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2012, 卷号: 109, 期号: 44, 页码: 18180-18185
作者:
Zhang, Xiaozhe
;
Wang, Jingjing
;
Feng, Yue
;
Ge, Jingpeng
;
Li, Wenfei
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
crystal structure
anion selection
cytoplasmic region
electrophysiology
single channel recording
Differential effects of activating D1 and D2 receptors on electrophysiology of neostriatal neurons in a rat model of Parkinson's disease induced by paraquat and maneb
期刊论文
NEUROSCIENCE RESEARCH, 2011, 卷号: 71, 期号: 4, 页码: 411-420
作者:
Xu, Haiyan
;
Chen, Ruirui
;
Cai, Xiaoyan
;
He, Defu
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
Neostriatum
Dopamine receptors
Parkinson's disease
In vivo
Electrophysiology
Crucial Points within the Pore as Determinants of K+ Channel Conductance and Gating
期刊论文
JOURNAL OF MOLECULAR BIOLOGY, 2011, 卷号: 411, 期号: 1, 页码: 27-35
作者:
Shi, Ning
;
Zeng, Weizhong
;
Ye, Sheng
;
Li, Yang
;
Jiang, Youxing
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
MthK K+ channel
steric hindrance
electrostatics
constriction point
single-channel electrophysiology
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